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    • Kinetic Optimization of Lysine-Targeting Covalent Inhibitors of HSP72. 

      Pettinger, J; Carter, M; Jones, K; Cheeseman, MD (2019-12-06)
      The covalent inhibition mechanism of action, which overcomes competition with high-affinity, high-abundance substrates of challenging protein targets, can deliver effective chemical probes and drugs. The success of this ...