Browsing Cancer Therapeutics by author "Knox, James"
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Lysine-targeting covalent inhibitors
Newton G; Knox, J; Newton, G (Institute of Cancer Research (University Of London), 2023-12-14)Targeted Covalent Inhibitors (TCIs) represent an increasingly important strategy in modern drug discovery. TCIs exploit high affinity, reversible ligands which are then modified with modestly-reactive electrophilic warheads ...